A novel synthesis of 5-functionalized oxazolidin-2-ones from enantiomerically pure 2-substituted N-[(R)-(+)-α-methylbenzyl]aziridines

  • Sim, TB
  • Kang, SH
  • Lee, KS
  • Lee, WK
  • Yun, H
  • 외 2명
Citations

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90

초록

5-Funtionalized enantiomerically pure oxazolidin-2-ones were prepared in one pot from commercially available chiral aziridines bearing an electron-withdrawing group at C-2 with retention of the configuration in high yields by regioselective aziridine ring-opening followed by intramolecular cyclization.

키워드

XYLOSE DERIVED OXAZOLIDIN-2-ONESCHIRAL AUXILIARIESEFFICIENT SYNTHESISSTEREOSELECTIVE-SYNTHESISASYMMETRIC-SYNTHESISDERIVATIVES3-ARYL-2-OXOOXAZOLIDINESANTIBACTERIALSAZIRIDINESINHIBITOR
제목
A novel synthesis of 5-functionalized oxazolidin-2-ones from enantiomerically pure 2-substituted N-[(R)-(+)-α-methylbenzyl]aziridines
저자
Sim, TBKang, SHLee, KSLee, WKYun, HDong, YKHa, HJ
DOI
10.1021/jo0261911
발행일
2003-01-10
유형
Article
저널명
Journal of Organic Chemistry
68
1
페이지
104 ~ 108