N-Methylative aziridine ring opening and asymmetric synthesis of MeBmt

  • Kim, Yongeun
  • Yoon, Doo-Ha
  • Ha, Hyun-Joon
  • Kang, Kyung Yeon
  • Lee, Won Koo
Citations

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초록

Asymmetric synthesis of MeBmt, an unusual amino acid constituent of cyclosporine A, was achieved from aziridine-(2R)-carboxaldehyde through highly stereoselective addition of (E)-crotylboronate and the subsequent N-methylative aziridine ring opening as key steps. (C) 2011 Elsevier Ltd. All rights reserved.

키워드

MeBmtAsymmetric synthesisAziridineRing openingCrotylationUNUSUAL AMINO-ACIDSTEREOSELECTIVE-SYNTHESISFORMAL SYNTHESISCHIRAL GLYCINECYCLOSPORINEALDEHYDESKETONES
제목
N-Methylative aziridine ring opening and asymmetric synthesis of MeBmt
저자
Kim, YongeunYoon, Doo-HaHa, Hyun-JoonKang, Kyung YeonLee, Won Koo
DOI
10.1016/j.tetlet.2011.08.048
발행일
2011-11-09
유형
Article
저널명
Tetrahedron Letters
52
45
페이지
5918 ~ 5920