An efficient synthesis of morpholin-2-one derivatives using glycolaldehyde dimer by the Ugi multicomponent reaction

  • Kim, YB
  • Choi, EH
  • Keum, G
  • Kang, SB
  • Lee, DH
  • 외 2명
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초록

[GRAPHICS] A new one-pot procedure for the efficient synthesis of novel 3-substituted morpholin-2-one-5-carboxamide derivatives using commercially available glycolaldehyde dimer as a bifunctional component with various alpha -amino acids and isocyanides by the Ugi five-center three-component reaction (U-5C-3CR) was developed.

키워드

SOLUTION-PHASE SYNTHESISARMSTRONGS CONVERTIBLE ISONITRILEALPHA-AMINO-ACIDS4-COMPONENT CONDENSATIONLIBRARIESISOCYANIDESPYRROLESALCOHOLSLACTAMSRESIN
제목
An efficient synthesis of morpholin-2-one derivatives using glycolaldehyde dimer by the Ugi multicomponent reaction
저자
Kim, YBChoi, EHKeum, GKang, SBLee, DHKoh, HYKim, YS
DOI
10.1021/ol016716w
발행일
2001-12-27
유형
Article
저널명
Organic Letters
3
26
페이지
4149 ~ 4152